Registration No.: PI/2004/VII/361/MP
Name: Kadam Rameshwar Uttamrao
Connect at: Linkedin
M.S.(Pharm.) Thesis Title:
in silico evaluation of P. aurigunosa LPxC Inhibitors
Research: 8
Kadam RU, Garg D and Roy N. Selective mapping of chemical space for Pseudomonas aeruginosa deacetylase LpxC inhibitory potential. Chemical Biology & Drug Design 2008, 71: 45-56.
Kadam RU, Kiran VM, Cordorio A, Ouaissi A and Roy N. Structure Function Analysis of Leishmania Sirtuin; an Ensemble of In Silico and Biochemical studies. Chemical Biology & Drug Design 2008, 71: 501-506.
Kadam RU, Chavan A and Roy N. Pharmacophoric features of P. aeruginosa deacetylase LpxC inhibitors: An electronic and structural analysis. Bioorganic & Medicinal Chemistry Letters 2007, 17: 861-868.
Kadam RU, Garg D, Chavan A and Roy N. Evaluation of Pseudomonas aeruginosa deacetylase LpxC inhibitory activity of dual PDE4-TNF α inhibitors: A multi-screening approach. Journal of Chemical Information and Modeling 2007, 47: 1188-1195.
Kadam RU, Garg D, Paul AT, Bhutani KK and Roy N. Evaluation of proinflammatory cytokine pathway inhibitors for p38 MAPK inhibitory potential. Journal of Medicinal Chemistry 2007, 50: 6337-6342.
Kadam RU, Shivange AV and Roy N. Escherichia coli versus Pseudomonas aeruginosa deacetylase LpxC inhibitors selectivity: surface and cavity-depth-based analysis. Journal of Chemical Information and Modeling 2007, 47: 1215-1224.
Kadam RU and Roy N. Cluster analysis and two-dimensional quantitative structure-activity relationship (2D-QSAR) of Pseudomonas aeruginosa deacetylase LpxC inhibitors. Bioorganic & Medicinal Chemistry Letters 2006, 16: 5136-5143.
Kadam RU, Kiran VM and Roy N. Comparative protein modeling and surface analysis of Leishmania sirtuin: A potential target for antileishmanial drug discovery. Bioorganic & Medicinal Chemistry Letters 2006, 16: 6013-6018.