Protein Name: | Muscarinic acetylcholine receptor M1 (P11229) |
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Gene Name: | CHRM1 |
Description: | |
PDB ID: | 5CXV |
Protein Family: | PF00001, PS00237 |
Protein Category: | Membrane Receptors |
This panel provides drug-protein interaction and their ADRs along with references
Interacting Drugs | Toxicity | Mechanism | Reference |
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Gabapentin | Anxiety | Significant adverse effects may occur through the interaction of the antidepressants with other receptors believed not to be related to the therapeutic action@ most importantly the muscarinic acetylcholine receptor (M)@ the histamine-1 (H1) receptor and the alpha-1 (alpha 1) adrenergic receptor@leading to anxiety [ ADR Type 2 ] | Cell-mediated side effects of psychopharmacological treatment |
Gabapentin | Nausea | Significant adverse effects may occur through the interaction of the antidepressants with other receptors believed not to be related to the therapeutic action@ most importantly the muscarinic acetylcholine receptor (M)@ the histamine-1 (H1) receptor and the alpha-1 (alpha 1) adrenergic receptor@leading to nausea. [ ADR Type 2 ] | Cell-mediated side effects of psychopharmacological treatment |
Gabapentin | Sleep Disturbances | Significant adverse effects may occur through the interaction of the antidepressants with other receptors believed not to be related to the therapeutic action@ most importantly the muscarinic acetylcholine receptor (M)@ the histamine-1 (H1) receptor and the alpha-1 (alpha 1) adrenergic receptor@leading to sleep disturbances. [ ADR Type 2 ] | Cell-mediated side effects of psychopharmacological treatment |
Masoprocol | Dry Mouth | Not Available | Large-scale prediction and testing of drug activity on side-effect targets |
Pirenzepine | Impair Working Memory | Blockade of hippocampal M2 muscarinic receptors impairs working memory performance of rats [ ADR Type 1 ] | Blockade of hippocampal M1 muscarinic receptors impairs working memory performance of rats |
Ritodrine | Hyperhidrosis | Not Available | Large-scale prediction and testing of drug activity on side-effect targets |
Ritodrine | Mental Disorder | Not Available | Large-scale prediction and testing of drug activity on side-effect targets |
This panel provides information on drug category